Utano, Gadziriro
"Neostigmine" (kwepfuti)
"Neostigmine" (majekiseni) iri chakaita zvokugadzirwa chinodhaka, huru vanoshingaira venhumbi anoita se neostigmine methylsulfate.
gadziriro iyi ane raidudzwa anticholinesterase basa, uye saka pashure kushandiswa kwayo anovandudza kuchinjwa excitation kubva tsinga kuti skeletal tsandanyama, nhengo dzomukati uye ziso kuatsanangura zvose cholinergic zvinokonzerwa, uyewo nokuti kunosimudzirwa gastrointestinal motility, anowedzera mataurire Árbol, dundira, kwemakemikari anobudiswa omumuviri uye secretion.
Kugadzirira "Neostigmine" rakapa kwete chete muchimiro mhinduro jekiseni, asiwo muchimiro mapiritsi, granules, izvo rinogadzira nomumukanwa kuturika (vana).
zvairatidza
Akati medicament rinoshandiswa pamberi myasthenia, nourema uye paresis, kusagadzikana gwenya basa pashure zvinokuvadza uropi, neuritis, encephalitis pashure, poriyo uye tuberculous yomumuzongoza.
Rinoshandiswawo kana kudiwa Mabatirwo optic tsinga atrophy, kuderedza intraocular nevamwe yemaziso rwuchiwanzwa, uye kana zvakakodzera constriction ari mudzidzi. In zvirwere izvi, kuti mushonga rinoshandiswa muchimiro samadonhwe ziso.
Rinoreva "Neostigmine" (majekiseni) rinoshandiswa kuti induction webasa, uye ane marwadzo nomugumisiro. Kazhinji mushonga inoshandiswa mukurapa, apo ikarapwa vachishandisa atony mudumbu, dundira uye bowel, rakundwa nomuromo.
Drug "Neostigmine" majekiseni, uyewo mamwe marudzi ari chinodhaka, rinoshandiswa chete nokuda inonyorwa, uye kubvumira zvirongwa zvayo akazvimirira aisanganisira wairambidza.
Kana mushonga rinoshandiswa nemuromo kwayo dose nokuti mukuru ari kubva ramazana kusvika namashanu hundredths magiramu uye vakaendeswa 3 kanomwe pazuva. Nokuti vana pasi pemakore gumi - mumwe kuzviuru a giremu nomumwe unozotevera gore, asi hapana zvinopfuura 0.01 magiramu pazuva.
Kugadzirira "Neostigmine" (majekiseni) anogona kupiwa zvose subcutaneously uye intramuscularly mune imwe mari 1 ml ane 0,05% mhinduro chinotarisirwa vana maererano chegumi Rine mamiririta pagore asi kwete kupfuura 0.75 milliliter, zvose akaita imwe kana mbiri nguva. The zvachose nguva kurapwa kunoenderana kwokuomerwa chirwere uye zvinogona kubva 15 kusvika 40 mazuva, uye mune zvimwe zviitiko kunyange refu.
Kana pane simba basa, mushonga "Neostigmine" (ampoules) rinofanira kushandiswa subcutaneous majekiseni , uye panguva imwe chete akatanga nzira "Atropine". Izvi zvinoitwa kamwe chete pakutanga kubvuma kana jekiseni. Uyewo, kuti mushonga chinotarisirwa nomuromo mune imwe mari 0,003 d ose 40 maminitsi 6 nguva, uye majekiseni akaita 0,05% mhinduro 2 nguva imwe awa muna 1.0 Rine mamiririta.
Kumunhu mukuru, kufadza zuva dose ndiyo 0,05 g, uye basa haafaniri kupfuudza nemashanu hundredths magiramu. Panyaya majekiseni, kufadza dose pazuva iri 0.006 g, rimwe dose vasina thousandths anopfuura maviri giremu.
Possible nemishonga
Pashure kushanda vakati Pfungwa kuonekwe bradycardia, manyoka, kuda kurutsa, kunoderedza BP, ikawanda Árbol secretion, simba uye neutachiona.
Kana munhu aiva manyoka uye abdominal marwadzo, uyewo kudira ziya, inoratidza imwe chepfu chaizvoizvo rinoreva "Neostigmine". zvinodhaka "Atropine" subcutaneously jekiseni muzviitiko izvozvo.
Haukwanisi kushandisa mishonga pamberi nepfari, yakawedzera tsandanyama matauriro, Árbol asima, angina, atherosclerosis, uye kusashivirira zvinodhaka ichi.
Drug "Neostigmine": wongororo
Pindura zvakanaka pakugadzirira ichi ndivo vanhu vanotambura myasthenia gravis, sezvazvakanyorwa kuitwa uchibatsirwa rusingaperi yokuzvigadzirisa mishonga.
Nhamba varwere kuti nzvimbo "Neostigmine" chinoreva zvakawanda kana vamwe vanozviita dzose majekiseni, nepo vamwe akarwawo kurishandisa chete neapo, uye vamwe havana kushivirira. Somunhu divi maturo, varwere vakawanda cherechedzai chimiro muromo yakaoma uye kunyanya salivation uye pfari.
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