UtanoKugadzirira

"Risperidon": mirayiridzo yekushandiswa. "Risperidone Organica": tsanangudzo, zvinyorwa, zvinopesana

Age, mupfungwa uye maitiro kuchinja zvinogona kuomesa upenyu kwete chete munhu anorwara zvikuru, asi yake denderedzwa yomukati. Mabatirwo psychogenic nezvimwe zvirwere muitiro wakaoma kunzwisisa, asi mushonga asingadi mira uye wekuvamba peri itsva aungazviita navo. Huru basa anopiwa kurapwa. Mahwendefa "Risperidone" analogs izvo izhinji kwazvo, vari pakati zvikuru nevanhu zvigadzirwa. Chii yavo rutivi? Sei kutora kwavari, uye kana vane chero contraindications? Ndinogona kushandisa mapiritsi aya kuti mwoyo? Mhinduro dzemibvunzo iyi tichaedza kupa munyaya ino.

Release chimiro uye sezvamunoita "Risperidone" chinodhaka

"Risperidone" Mahwendefa zvinoberekwa makambani akawanda mishonga pasi chete zita uye vane substantially chete nziyo. The chikuru vanoshingaira wemafuta mushonga chaizvoizvo pacharo risperidone mune imwe mari 1, 2 kana 4 MG (zvichienderana chipimo chemushonga). Hwendefa Mumwe zvinenge zvakazara enteric-zvemapuranga Kamudzira chena. hwendefa iri kumativi, biconvex. In muchinjikwa-chikamu chinoratidza zvakajeka akaturikidzana maviri: wokunze uye yomukati. The Zvinoumba mahwendefa "Risperidone" - kuwedzera basa chirungiso - anowedzera zvinoriumba: starch, nesilicon dioxide, magnesium stearate uye MCC.

Mahwendefa "Risperidone" uye avo analogs, kusanganisira "Risperidone Organics", vakaradzikwa pepa Mabhokisi 10 zvidimbu mumwe izvo, akavapindurawo, akaisa mumabhokisi makadhibhokisi 2, 3, 5 kana 6 packs it pamwe chete mirayiridzo kushanda. Kuwedzera chigadzirwa zvinogadzirwa uye mumidziyo yose murima negirazi, nerimwe iro ringave riine mahwendefa 20, 30, 50 kana 60. Banks uyewo inoiswa mumabhokisi makadhibhokisi nemirayiridzo.

mushonga sei?

The kuitika "Risperidone" mapiritsi fuma kurairirwa chokuita bensizoksazola, kureva neuroleptics. Kuwedzera kune antipsychotic mugumisiro zvinodhaka ichi ane kunyaradza, hypothermic uye antiemetic zvivako. Izvi imhaka kukwanisa adzikatidza tichishingaira chirungiso D2-receptors muna Mesocortical uye mesolimbic hurongwa uye emetic nepakati, uye kukanganisa adrenergic receptors vemunyika muuropi hunde. Uyewo mukomboni anokwanisa kuvhara dopamine receptors ari hypothalamus.

Nokuda akadaro pharmacological ehupfumi zvinodhaka "Risperidone" ratings iyo inenge nguva zvakanaka, anokwanisa kudzvinyirira zviratidzo neurogenic zvirwere zvakadai zvinovadadira uye fungidziro, utsinye uye automaticity. Against ichi nechekumashure, nyanzvi dzinoti kuti mushonga une anenge hapana zvazvinoita gwenya basa, asi panguva imwe chete, anovanza symptomatic kuvhiringidzika zviratidzo schizophrenia.

Distribution uye excretion

The kuitwa yezviri fuma iri nemudumbu kunoitika munguva pfupi nguva uye kune kunonyanyisa papi. Food yaunodya hazvirevi vliyaetetot rikurumidze. Maximum wakafananidzwa ari plasma vanoshingaira mumiririri rinosvika paawa pashure achitora zvinodhaka. Dérivés sezvo risperidone (9-hydroxyrisperidone) vari kunyura zvishoma nezvishoma.

Nezveshoko kuparadzira zvinodhaka mumuviri "Risperidone" mirayiridzo Chinyorwa anoti pamusoro kupinda yezviri fuma iri munyama siyana uye nhengo, uye uropi, uye mukaka. Kukurukura mapuroteni eplasma hazvisi vanenge 90%.

Hafu-upenyu zvinodhaka kunoitika mumatanho maviri: mumaawa 3 pedo 70% of mukomboni yabudiswa kubudikidza itsvo dziri kuchinja chimiro, nepo 9-digidrorisperidon akaratidza anenge pazuva. Varwere vakwegura uye vaya vanotambura itsvo kukundikana, nguva excretion zvinodhaka yakawedzera.

Kushandisa zvinodhaka: zvairatidza uye contraindications

Shandisa rinorumbidza zvinodhaka "Risperidone" mirayiridzo Chinyorwa kuti kana zvinotevera zvirwere kana zvinetso mumuviri:

  1. Chenjera kana chirwere muchimiro schizophrenia.
  2. Psychopathic nyonganyonga, dzinoratidzwa kunaka kana zvibereko symptomatic kuratidzwa.
  3. Mental chirwere, achiperekedzwa zvinyamusi.
  4. Dementia Kazhinji chinoita panomuka hasha uye utsinye, zvinovadadira uye dzimwe pfungwa zviratidzo.

Also kuratidzwa ndiye chinodhaka "Risperidone" vana vavo vari kuyaruka vane nzvimbo chirwere (dzinoparadza pfungwa) vanoziva remangwana kana zvinofunga kana nepfungwa retardation, uyewo nedambudziko zvirwere uye zvokudarikidza zvakasiyana. Muzviitiko izvi, hwendefa wakakurira kutsigira basa iri kurapwa.

It chiri zvinodhaka uye kukosha contraindications anosanganisira hypersensitivity kuti zvinoumba mahwendefa. Mukuwedzera, zvinodhaka "Risperidone" mirayiridzo Chinyorwa rinokurudzira kushandisa nokungwarira kunyanyisa mune zvinotevera zvirwere kana mamiriro:

  • uropi namamota uye ropa riyerere chepfungwa;
  • hepatic uye renal kukundikana kwazvo chimiro;
  • Zvirwere intestinal patency;
  • mwoyo chirwere, kusanganisira myocardial infarction, mwoyo kukundikana, chisingaperi chimiro antrioventikulyarnaya nechigumbuso uye bradycardia;
  • Drug ovhadhozi kana kuvimba navo;
  • kupera muviri;
  • Parkinson nehosha;
  • chinyamunhari chinorwadza (panguva zvinodhaka kana chirwere);
  • Pamuviri uye lactation.

Uyezve, mushonga hauna varumbidzwa "Risperidone" (Mahwendefa) iri kuora mwoyo, izvo kwakunoitwa rutapudzo murwere basa uye vachida kuzviuraya. Uyewo nokungwarira prescribers vanhu vane zera harina asvika makore 15.

Chipimo chemushonga uye nzira kugamuchirwa

Chipimo chemushonga uye nzira kuvimba mushonga anowanikwa pakaunda murwere chirwere, kukuvadza ari vhinza, uye kuvapo concomitant zvirwere kana pathological inoti. All akakodzera mashoko pamusoro kushandiswa zvinodhaka "Risperidone" unogona kuona tafura.

Chirwere kana ezvinhu

chipimo chemushonga

Application Notes

schizophrenia

Kutanga dose - 1 MG 2 kanomwe pazuva. Dose muna 2nd uye mazuva hunotevedzana ndiyo 4 MG (2 MG 2 kanomwe pazuva).

Kana mushonga "Risperidone" anogadzwa somutsivi womutariri zvimwe zvinodhaka, yezwi rinofanira kuitwa zvishoma nezvishoma.

Dementia nezvimwe zera naresheniya

1 MG pazuva, kutora mushonga inofanira kuva 1 nguva pazuva.

In pamberi nenyonganiso ose itsvo nerevane chiropa dose kuderedzwa 2 nguva, zvishoma nezvishoma kuwedzera kusvikira inokurudzirwa.

Kukara, nedambudziko kana zvimwe zvirwere zvepfungwa

Kutanga dose - 2 MG pazuva (rimwe zuva muna mabiko), ipapo dose iri kuwedzera zvishoma nezvishoma kusvika 6 MG pazuva.

Ndapota varangarire penguva pakati dose inowedzera of 2 mazuva.

Maitiro asina kutsarukana muna kuyaruka

1 MG pazuva, vasina kugamuchira

uremu murwere hakufaniri kuva makirogiramu asingasviki 50, vakomana kana chipimo chemushonga anofanira kugadziriswa.

Mental retardation iri pakanyorwa zvinoparadza chirwere chepfungwa

1 MG pazuva

Kana chinokosha mukana zvokudarikidza uye inodiwa rutapudzo gipermany kwokutanga dose pamwe zvishoma nezvishoma nokuwedzera kusvika kunokurudzirwa.

haafaniri kupfuudza 16 MG upi chirwere kana ezvinhu daily dose "Risperidone" gadziriro.

Nenjodzi yacho Muviri ovhadhozi

Chimwe chinokosha kuti unofanira kuziva varwere anozadziswa nzira yokurapa ne "Risperidone" - nemishonga kuti zvingaitika munguva nedanho negashiro pamahwendefa. The ndingangokuvara chiitiko kwavo kunoenderana achinyanya pamunhu. Saka, chii chinogona kunokanganisa murwere?

Most dzichitaridzika zvinotevera nenjodzi kubva siyana nadzo uye nehurongwa:

  • Zvirwere vaikudzwa kufema uye Urinary turakiti (kunyanya varwere vakwegura chirwere kuti "Dementia");
  • nomusoro, nenyonganiso kuti hope, dzungu, hope uye madzerere;
  • dyspepsia, epigastric kurwadziwa, kuda kurutsa, muromo yakaoma;
  • mwoyo mutinhimira zvirwere (tachycardia);
  • edema of nasal mucosa uye Eustachian chubhu apo murwere anonzwa stuffy mhino kana nzeve, mhino bleeds;
  • chikosoro, runny mhuno, uye kupfupika mweya;
  • kupererwa neropa;
  • Urinary incontinence;
  • kuzvimba majoini, kuchinja gait (kunyanya varwere vakwegura), shure marwadzo uye kurwadza kwemajoini.

kunewo vakawanda nemishonga, izvo panongova kashoma kuitika mu "Risperidone" achitora mushonga. Reviews Nyanzvi dzinotaura pakati pavo zvinotevera:

  • nzeve uye ziso zvirwere;
  • kutapukirwa noutachiona kukanganisa muviri wose kana vemunyika;
  • kufema turakiti zvirwere, kusanganisira mabayo, tonsillitis, bronchitis uye tracheobronchitis;
  • onychomycosis uye acrodermatitis;
  • kuvhiringidzika, kufunganya, zvokudarikidza uye hypomania, dyskinesia;
  • Tsandanyama Rigidity, hyperthermia, vakawedzera vangadikitira;
  • kusagadzikana oscillations BP;
  • pfari;
  • kufema, yokumusoro yemweya occlusion sputum (miridzo panguva afemeruke, manyoro rales kana dysphonia);
  • kuwedzera kana kudzikisa uremu;
  • kumwedzi hadzina kufambiswa zvakanaka, kushaya ejaculation, priapism, kushaya chido chokurara;
  • zamu soreness kuti tsandanyama;
  • kuzvimba ganda, kunyanya chiso, chills, nyota, yokuSpain-kufanana nehurumende;
  • kusimba maoko nemakumbo, kunzwa zviri kuomarara majoini.

Kana chakakomba kukunakira kuti kutora zvinodhaka "Risperidone" anoreva zvakafanana zvinodhaka angasava chakakodzera amirire mishonga, sezvo ane chete unorapa. Panyaya iyi, nyanzvi achasarudza mumwe mushonga, iro rinoumbwa mamwe yeimwe, kana kupa mamwe mishonga kubvisa hachifadzi zviratidzo.

Zviratidzo uye mabatiro zvinodhaka ovhadhozi

Kana mirayiridzo kukodzera dosages kumusoro mudenga ovhadhozi zvingaitika, iyo inotaurwa iziviswe uye kuramba richikwidibira ropa dzvinyiriro uye mwoyo mutinhimira zvirwere (tachycardia). Mukuwedzera, murwere anogona kanganisa somnolence, nyaradzo, kufema zvirwere uye extrapyramidal nyonganyonga.

Dzakananga mushonga mukugadzirwa "Risperidone" kwete, saka kurapwa nechinangwa kubvisa kupfuura akazivisa zviratidzo. Sezvo rubatsiro wokutanga murwere zvinofanira kusukwa dumbu uye kupa neactivated charcoal uye laxatives. Akaroromesawo BP mitemo yakaoma zvinoda intravenous kwokubatsira agonists uye aizomupa mhinduro.

Mumazana nguva inodiwa cardiac zvichiongororwa kuziva nekuve cardiac arrhythmias. Kana paine aonekwa, mishonga mishonga yakakodzera.

Mirayiridzo kushandiswa kwezvinodhaka

Kana muchigamuchira zvinodhaka "Risperidone" mirayiridzo Chinyorwa rinokurudzira kutevera mashoma mirayiridzo inokosha. Izvi zvichaita kwete chete kuderedza mukana wokuti nemishonga, asiwo kuvandudza zvinonyatsorehwa ezvinhu omurwere pamberi co-morbidities.

Chokutanga iwe uchida mari Cherechedzai chipimo chemushonga zvinodhaka kune varwere maari pane zvirwere kumwoyo. Panyaya iyi, kutanga kugamuchira zvinodhaka zvakafanira shoma mishonga, zvishoma nezvishoma vachiwedzera kuti vaida tsika. The chete mazano anoshanda panyaya hypovolemia, kupera muviri uye cerebrovascular zvirwere.

Nyanzvi vanotiwo varegedze pakushandisa mukuru-mafuta zvokudya uye Kudyisa sezvo vakadaro. Izvi imhaka yokuti mishonga zvinodhaka "risperidone" refu ndingangokuvara kutaridza mamwe uremu.

Hazvina varumbidzwa panguva kurapwa mapiritsi "Risperidone" kuita zvinhu zvine chokuita basa motokari nezvimwe zvigadziriswe kuti zvinoda yakakwirira pfungwa murwere uye nokukurumidza psychomotor zvavaifunga.

Kudyidzana nevamwe zvinodhaka

In agadza zvinodhaka "Risperidone", mitengo yakanga dzichakurukurwa Papera, vanofanira kufunga kugona yayo kutaura zvakawanda nemishonga. Mune zvimwe zviitiko, izvi zvinogona kutungamirira isingatarisirwi uye kwete inofadza chaizvo zvaitika. Saka, zvinodhaka, mwoyo chaizvo huta yevanhu hurongwa, uyewo panyaya iyi, pamwe chete "Risperidone" kumutsa ezvinhu akadai, ive chirungiso CNS mwoyo mabasa.

Vamwe zvinodhaka, zvakadai Beta-blockers, vazhinji, zvose, pasina chaakasiya tricyclic antidepressants anogona kuwedzera wevasungwa yezviri fuma "Risperidone" mahwendefa plasma. The Ndozvakaitawo mushonga "Fluoxetine". "Carbamazepine" nekusiyana, akazoita wevasungwa kuti vanoshingaira fuma rinoreva "Risperidone" plasma. At kugadzwa kwavo vadyi kunoda kuramba zvichiongororwa murwere, uyewo kuchinja ari dosing zvaiitwa.

Reviews

Reviews zvemahwendefa "Risperidone Organics" uye "Risperidone", mutengo uko kuonekwa nyore zvakawanda vatengi (avhareji 170 rubles por rongedza), hazvigoni kunzi kunaka. Kuvhiringidzwa kuti mahwendefa hosha dzakasiyana-siyana psychogenic kana zvounhu, akanaka maonero zvose nyanzvi uye varwere. Just norudaviro uye analogs zvinodhaka ichi, nekuti kakawanda kusiyana maviri chete mari uye Zvinoumba anongoda chete (kunze Excipients).

The chete kuchikosha drawback Mahwendefa "Risperidone" (analogs pamusoro vanoshingaira zvinhu vachawa pasi tsanangudzo iyi) - yakawanda nemishonga, izvo dzimwe nguva zvingaita unhu murwere upenyu huve nani. Ndokusaka nyanzvi dzinokurudzira panguva panowanikwa chero nenjodzi kubata chiremba wako kugoverana naye kuwana nzira kubva izvi.

Saka takadzidza kuti dzinomiririra "Risperidone" mapiritsi. Instructions, mutengo, analogs uye nenjodzi dzomuviri zvadzidzwa pepa rino zvakadzama. In mhedziso, ndinoda kukuyeuchidzai kuti mushonga asunungurwa chete mushonga. Kunze komutemo basa uye nokugamuchira mahwendefa boka iri angava utano hwako.

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