Utano, Gadziriro
The mushonga "tizanidine": mirayiridzo kushandiswa, anofanana. "Tizanidine-din email", "tizanidine-Ratiopharm"
Chii dosages ramakanzi zvinodhaka "tizanidine?" Mirayiridzo kushandiswa medicament rinotaurwa hereinafter. Uyewo, kubva zvinhu ino uchadzidza pamusoro mune fomu rinobudiswa, yakati rinoreva kuti chikamu chacho, kana ane marwadzo, uye contraindications dzomuzana.
The chimiro, description, akafanana
Chii murwiyo rine mushonga "tizanidine?" Mirayiridzo Dzokushandisa inoti yezviri chezvinonhuwira kwezvinodhaka izvi tizanidine. Uyewo nemamiriro vaiona medicament unotora sezvo Excipients lactose anhydrous, colloidal nesilicon dioxide, microcrystalline cellulose uye stearic acid.
Drug "tizanidine," iyo mirayiridzo midzi muna atorwa, akaita muchimiro mahwendefa kumativi chena. Kune rimwe divi panoparadzana ubvise ndiye chinodhaka, uye wechipiri - ndezve kuti T4 uye T2.
pharmacological zvinhu
Chii mashandiro chiito "tizanidine" chinodhaka? Mirayiridzo dzokushandisa kunoratidza kuti mhasuru relaxant. Pashure pokugamuchira Mahwendefa mukati zvinodhaka vanoshingaira fuma kunoderedza skeletal tsandanyama tonus, richikwidibira kurwisa kwavo pusa inofamba uye deceleration pamusoro spasmodic siyana uye enhancement pamusoro zvemasanga zvazvingava.
Kubva pane zvataurwa zvinganzi nyore kucherechedzwa kuti vaiona zvinodhaka inosimudzira tsandanyama-vakazorora kushanda. Izvi zvinoitika nokuda kwokudzvinyirirwa polisinapticheskie musana hunenge. Izvi zvakafanira nokubudiswa amino acids kubva zviteshi (presynaptic) kuti musana interneurons.
pharmacokinetic parameters
Ndezvipi pharmacokinetic parameters ane zvinodhaka "tizanidine" (Mahwendefa)? Mirayiridzo kushandiswa munyaya iyi anopa nzwisisika ruzivo.
Pashure zvokuudzwa kwokubatsira ari medicament wefodya chose. bioavailability Its Mhedziso anenge 40% (nokuda zvikuru rokutanga nomunyika chiropa).
The rinoita mushonga fuma iri kuparadzirwa vose hurongwa uye munyama. kwawaiitwa pamwe mapuroteni kweinenge 30%.
The hafu-upenyu zvinodhaka ndiko maawa 2,5. About 95% of dose rinoita. Akaratidza medicament kuburikidza itsvo (vanenge 60%) nemudumbu (vanenge 20%).
zvairatidza
Mune zvimwe zviitiko, akarayira kuti zvinodhaka "tizanidine?" Kushandiswa mishonga iyi zvinonyatsoshanda mune spastic mamiriro skeletal tsandanyama, kunoitika apo chetsinga zvirwere zvakadai:
- Kurohwa;
- chinopedza musana chirwere;
- chisingaperi myelopathy;
- nemultiple sclerosis.
Uyewo mushonga "tizanidine" kuratidzwa panguva kurwadziwa ari tsandanyama, izvo kuva nokuda kukundwa vari nomuzongoza.
Contraindications
The huru uye zvichida chete contraindication zvinodhaka ichi ichiwedzerwa murwere aikanganiswa tizanidine. Uyewo, zviri rambidzwa kutora pachiimbwa nzira dzakadai se "Ciprofloxacin" uye "Fluvoxamine".
Drug "tizanidine": mirayiridzo kushandiswa
Maererano mirayiridzo, kwokutanga chipimo chemushonga "tizanidine" medicament ndiyo 2 MG.
Sezvo kubata zvinodhaka zvasvika rinozotora maawa 1-2 uye rakasanganiswa pashure pemaawa 3-6, mishonga yaifanira pa zvikamu maawa 6-8. Saka, panguva zuva havachiri pane 3 Mahwendefa.
The chipimo chemushonga pamusoro medicament iri kuwedzera zvishoma nezvishoma kusvika 4 MG (pa dose). Zvisinei, kuita kudaro chete kuna kana, pashure 4 mazuva kurapwa mugumisiro haina akaratidza.
Vose daily chipimo chemushonga zvinodhaka hakufaniri kupfuura 36 MG. Panyaya chipimo chemushonga zviumbu, negashiro vanopfuura 16 MG kuti vanachiremba harina kudzidza.
- In renal insufficiency. With ichi chirwere mapiritsi ushandiswe nokungwarira zvikuru.
- Abnormalities mu chiropa chaitika. Drug "tizanidine" kungwarira pachii vanhu vane chero chiropa kukundikana. In varwere izvi, munhu wacho chipimo chemushonga anofanira kuderedzwa. Zvakakodzera kuramba kuongorora padanho aminotransferase. Wokutanga zvichiongororwa akaita mwedzi mumwe pashure mharuro kurapwa.
zviitiko ovhadhozi
Clinical zviratidzo kuitika tikafunga ovhadhozi vangava zvakasiyana zvachose pharmacology. Kazhinji, varwere vane lethargy, kuvhiringidzika, hope uye pakoma. Mukuwedzera, mushonga pamatunhu mishonga inogona kukonzera dysfunction mwoyo tsandanyama, kusanganisira panowanikwa bradycardia uye hypotension.
nemishonga
Pane divi migumisiro Varwere pakugamuchira "tizanidine" chinodhaka? Mirayiridzo yokushandisa (anoreva zvakafanana pamusoro chishandiso zvinoratidzwa hereinafter) rinoti kuti nyaya medicament kunogona kukonzera muromo yakaoma, hope, hypotension, bradycardia, kuderera BP, dzungu, tsandanyama chinyamunhari chinorwadza, kurukutika, utera, kurukutika, kuvhumuka, hepatotoxicity, kusagadzikana chiropa.
Very kashoma kubatwa zvinodhaka izvi zvinosimudzira chitarisiko Stevens-Johnson urwere, exfoliative dermatitis, anaphylactic kuvhunduka, ventricular tachycardia, hepatitis, kuora mwoyo, nezvipusha, kurwadza kwemajoini, mapundu, paraesthesia uye tremor.
zvinodhaka kwavatori
Asati kushandisa "tizanidine" chinodhaka vanofanira kuverenga kunyatsoongorora mirayiridzo. Rinoti zvinotevera zviri zvayo zvinodhaka mukukurukurirana:
- Akabatana "ciprofloxacin" uye "Fluvoxamine" anogona yekudyidzana kuderera BP, uye kutanga hope. Uyezve, kugadzirira kunzwisisa kwakadaro kunopesana hwevanhu psychomotor mabasa.
- Mawa kurapwa nemishonga pamwe CYP1A2 FIs (semuenzaniso, "zileuton" "Fluoroquinolones", "Amiodarone", "Mexiletine", "propafenone" "Verapamil," "Cimetidine" "Famotidine" "acyclovir" uye "ticlopidine") zvakasimba contraindicated.
- Not akakurudzira mapiritsi zvabatanidzwa "tizanidine" pamwe nemumuromo pamuviri. Kana mamiriro murwere zvinoda mawa yaitonga mishonga iyi, kutanga dose inofanira kuva shoma. Negashiro dzakakwirira mishonga zvinodhaka kungaita kuti nemishonga yakadai hypotension, bradycardia uye hypersomnia.
- Sangana mushonga uyu doro haisi inokurudzirwa. Izvi imhaka yokuti doro kunowedzera wevasungwa yezviri zvinodhaka fuma muropa, uye izvi zvingaita kuti vasingadiwi migumisiro.
pasherufu upenyu, okuchengetera uye kutengeswa mamiriro
Mahwendefa "tizanidine" kupiwa mu Pharmacies pamusoro chiremba mushonga. Vanofanira zvinganaka ane mumupanda tembiricha munzvimbo ine rima. Zvakafanira kudzivirira mushonga kubva kuvana vaduku.
Pasherufu upenyu mari ndiyo 3 years. Pashure iyi nayo hakubvumidzwi kutora.
Price, anoreva zvakafanana uye analogues zvinodhaka
Mishonga yakasiyana akadai "tizanidine," "tizanidine Ratiopharm" uye "din email tizanidine?" Mirayiridzo kushandisa nzira idzi rine chete zviratidzo, marwadzo, contraindications, nzira chourongwa uye dosages. Musiyano chete pakati anotaurwa mishonga vagadziri dzavo. Saka, vose mari izvi anogona kunzi anofanana.
Kana rakasiyana "tizanidine" chinodhaka, ipapo vanosanganisira zvinodhaka zvakadai se "Sirdalud", "Tizalud" uye "Sirdalud MP."
How zvikuru ndivo "tizanidine," "tizanidine din email" uye "tizanidine Ratiopharm"? The Mirayiro yakatora zvinodhaka izvi, asingadi kupindura mubvunzo. Kuziva mutengo nzira idzi ukangogamuchira kukwanisa kurwisa. Kazhinji, hazvina yakakwirira chaizvo uye anenge 120-170 rubles Russian (zvichienderana neuwandu mapiritsi ari pasuru uye mugadziri).
Zvinofanira pakarepo kucherechedzwa kuti medicament "tizanidine" ane hwakanyatsorwisa chipa mari (somuenzaniso, analogs akadai "Sirdalud", "Tizalud" uye "Sirdalud MR" vari zvishoma anodhura, vanenge 240-270 rubles). Ndokusaka varwere vakawanda zvatinofarira yavo yokutanga zvinodhaka.
mishonga Reviews
Zvino munoziva sei kushandisa mishonga yakadaro "tizanidine," "tizanidine Ratiopharm" uye "din email tizanidine." User kubvuma nevamiririri izvi kwave kukurukurwa pamusoro.
Varwere vanenge nokusingaperi akashandisa mushonga uyu, muende munzira dzakasiyana-siyana. Vazhinji wongororo kuti zvinoita kugumisa kuti mushonga "tizanidine" haugari kusangana zvomurayiro varwere.
Vanhu vazhinji vanoti kuti zvinodhaka izvi rimwe nyaya matatu kukonzera marwadzo akadai kwazvo chinyamunhari chinorwadza uye tsandanyama pari. Similar kuitike pakarepo pashure pokushandisa medicament.
Pashure kushandisa wechipiri mapiritsi, vamwe varwere vanonzwa simba, nzwa dzungu, uye shungu kukurutsai. Kana zviratidzo zvakadaro, nyanzvi dzinokurudzira kuti kurega kugamuchira mari, kana kusimba ravo zvowedzera.
Mune zvimwe zviitiko, pashure kushandisa "tizanidine" vanhu vane matambudziko dzvinyiriro uye dumbu, uye mwoyo palpitations.
Zvinofanira kucherechedzwa kuti nyaya dzinovaka kubva mushonga pasi pakudzokorora haisi zvokuti. Pakati pavo vane kuvapo uye yakaderera Mari zvinodhaka.
Tichifunga zviri pamusoro apa zvinofanira vakagumisa kuti kutora mishonga "tizanidine" uye ayo anoreva zvakafanana, chete kuti sezvinoratidzwa uye chete mushonga.
Tichifunga vakawanda nenjodzi, nyanzvi haisi yakarumbidza kushandisa zvinodhaka panguva yepamuviri uye panguva uchiyamwisa, zvikasadaro zvingava anokanganisa utano mwana kana mudumbu.
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