Utano, Gadziriro
"Betacam": mirayiridzo kushandiswa, analogs uye wongororo
Kubvisa dzakakwirira kumanikidzwa uye siyana cardiac zvirwere vachishandisa beta1 adrenoblokatornye nzira. Imwe mishonga yakadaro zvinodhaka "Betacam". Mirayiridzo kushandiswa se mushonga kuti rinoratidza cardioselective, antihypertensive uye sympathomimetic chiito.
unhu zvakafanana
chokushandisa ichi anonzi chakaita zvokugadzirwa beta1-adrenergic blocker. Yakabudiswa neZvapupu Kupro chirimwa "Medokemi LTD" iri Hwendefa muchimiro ane chena kana substantially chena unhani mumuhara.
Medicament "Betacam" mirayiridzo rondedzero rekugadzirira rine marudzi anotevera: vane woita chimiro pamwe biconvex hukawanika, pane Kuparadzaniswa ubvise ngozi. Kana iwe kuputsa upi piritsi, ipapo ichava zviri yomukati chena kana anenge chena.
On medicament "Betacam" mirayiridzo mutengi pasuru tsananguro zvipo zvinotevera nzira: mumwe rongedza rine Maronda akasiyana matatu. Mumwe gandiwa Sero ndiro riri mumapepa ari pamahwendefa 10.
mamiriro
In mushonga mukuru basa kunopiwa magetsi pakuderedza muchimiro betaxolol hydrochloride munyu. The chipimo chemushonga rimwe piritsi iri 0,020 d
A achishandisa "Betacam" mirayiridzo iri Zvinoumba vakaneta zvinhu zvinorondedzerwa pasina chaiyo nhamba yavo. Mahwendefa akaumba starchy yavaibvisa glycolate, shuga, mukaka, magnesium stearate, microcrystalline cellulose mhando, aerosil, titanium oxide, uye polyethylene glycol hydroxymethylpropylcellulose chiratidzo 400.
mashandiro chiito
On mushonga "Betacam" mirayiridzo Chinyorwa inosimbisa cardioselective beta1 -adrenoblokatornuyu pasina mukati sympathomimetic basa simba. Mahwendefa kuratidza murombo Kamudzira pakudzikamisa kushanda.
Antihypertensive basa iri nokuda zviito kuti kuderedza cardiac goho mwoyo tsandanyama uye kuderedza tsitsi dzishande muropa midziyo panguva arikunze.
Selectivity Migumisiro zvinodhaka riri paumbwe β 1 -adrenoreceptor haagoni kunzi isiyo, nekuti yakakwirira mishonga pamusoro betaxolol ingachinja β 2 Kanotokonya -adrenozavisimye inotungamirwa izvo dziri muna principales uye ropa midziyo.
Ichivharira Zvakaitwa chinodhaka, kufungisisa pharmacodynamic unhu chokuita vasanyanye kwemwoyo panguva yokuzorora uye panguva yechiitwa. Zviri nokuda chinovhiringidza kuti β-adrenoceptor idzodzo dziri sinus raiva pedyo nebundu, izvo DZEMUNHU DZINODZORA automaticity yavo.
It kunoderedza kusunungurwa myocardial hunoshamisa mune basa uye pusa ezvinhu muviri, izvo zviri kukonzerwa yemakwikwi daka pakati catecholamines uye peripheral tsinga harinzwi pakati adrenergic mhando.
The mushonga kunoita systolic uye diastolic BP iri arteries pakuzorora uye panguva yechiitwa, kunoderedza dzepanguva orthostatic kuwedzera kakawanda mwoyo sunga. Zvakadaro zvakaitika zvinodhaka kunoderedza mutoro pamusoro myocardium.
Beta adrenoblokatornoe zvinoreva rine antihypertensive webasa anotevera mashandiro:
- ungaderedza cardiac goho;
- yakapedza spasm ari tsinga panguva arikunze nokuda nechepakati chiito, izvo ichikutadzisa kurova kwemwoyo tsitsi kune vascular masvingo panguva braking renin basa.
Yakareba kwokubatsira mushonga hazvideredzi ayo vane chirwere cheBP maturo. Kana tikatora rimwe dose betaxolol 0,005 kana 0,04 g, kumanikidza rutapudzo vacharatidza chete pashure 3 kana 4 awa.
Mukurapa, "Betacam" User Application kunoratidza kuti kutungamirira munhu chipimo chemushonga 0.005g chikonzero antihypertensive mugumisiro ane kuchinyanya kakapetwa maviri kudzika pane pamwe yose piritsi.
Kufadza antihypertensive basa chero wevasungwa ose betaxolol rinowanika pashure pemazuva 7-14.
Kuchirapa dosages ose medicament regai kukonzera akasiyana cardiodepressivny Chaizvoizvo, hapana zvazvinoita shuga muviri, kunonoka asingadi kuwedzera yavaibvisa cations uye mvura munyama.
Chii rinoshandiswa
Drug "Betacam" mirayiridzo yechipupuriro chinosanganisira zvinotevera mitsetse:
- cheBP;
- coronary tsinga chirwere myocardial hunoshamisa tsandanyama, myocardium infarction pakuitika;
- hypertrophic cardiomyopathy.
The mushonga ushandiswe kana paine kuchinja mwoyo, varehwa ari kumhanyisa iri sinus mutinhimira, ventricular tachyarrhythmias uye supraventricular hunhu, kunonoka depolarization pamusoro myocardium, arrhythmia chokuita prolapse mu mitral vharafu, kunyanya kugadzirwa thyroid mahormone.
How kushandisa
On mushonga "Betacam" mirayiridzo kushandiswa pendi dose zvichienderana murwere ezvinhu. All daily dose drink pa kunwa. Food haadi kukanganisa Absorção de Água kurapwa. Hwendefa zvinofanira kusukwa pasi nemvura yakachena.
Inosimudzira BP kubatwa daily pokutangira dose inobva 0,005 kusvika 0,010 d Pashure 7 kana 14 days, kana zvakakodzera, kuti kuwedzera uwandu medicament 0,020 d
Ndiani havafaniri kushandisa
Haasi munhu wose kunoita kushandisa nzira "Betacam" mirayiridzo Chinyorwa. Contraindications chokuita kunyanya aikanganiswa zvokubikisa, uyewo betaxolol hydrochloride.
It haungopiwi varwere vane chirwere mwoyo tsandanyama insufficiency nezvimiro sinoatrialnuyu uye atrioventricular blockage ari dhigirii wechipiri nowechitatu, bradycardia, hypotension, Árbol asthmatic kurwisa, vaingoerekana angina.
Zvinodhaka "Betacam" Mahwendefa mirayiridzo kushandiswa vari haana varumbidzwa drink mhando pamwe cardiogenic kuvhunduka, vascular angiotrofonevroze magumo, kuwedzera tsandanyama myocardial hunoshamisa, asthenic ophthalmoplegia, endarteritis obliterans, emfizemnom lesion pamusoro zvemapapu rinenge chisingaperi obstructive bronchitis unhu chirwere cheshuga mellitus.
Pachena kuchinja itsvo psoriatic maronda iri contraindicated kuti kurapwa.
nenjodzi
Nemigumisiro rinoreva "Betacam" User zvikumbiro zvinosanganisira anonoke kurova kwehana, atrioventricular blockage, cardiac tsandanyama insufficiency, orthostatic donhwe kumanikidzwa, murombo kuparadzirwa vakapoteredza arikunze, maoko kazhinji chando uye netsoka, paresthesia. Saka kwakakanganiswa vascular maitiro uye mwoyo.
Árbol spasm, mapundu, urticaria, psoriasis, yakaoma ziso mucous Kamudzira zvingaitika divi siyana uye kufema ziso zvomukati, ganda.
The mushonga anogona kukonzera hope, asthenic ezvinhu, zvokuora mwoyo, kunyanya kuneta, kuvhiringidzika, zviratidzo zvisipo, nzwa dzungu uye kutemwa kurwadziwa.
Zvisingadiwi pezvakaitwa ari zvomudumbu ino dzinoitwa kuda kurutsa, retching, manyoka, kunonoka cheya cholestasis.
Other kuratidzwa zvinodhaka chiito aigona kuva kuderera kuti leukocyte uye masero platelet ropa, uye dzikira potency.
Features kurapwa
Kubvuma chero mushonga vangava chokuita nedzimwe nuances, izvo kuvimba pharmacological mapoka, murwiyo uye chipimo chemushonga zvinodhaka kushandiswa.
Mishonga "Betacam" mirayiridzo kushandiswa mirayiridzo inokosha vanopiwa neimwe nyaya dzisiri mureza, inoda kugadziriswa.
Saka panguva Danho rokutanga kurapwa kunogona kukonzera kushaya mwoyo tsandanyama vanhu asingatani kutsauka ichi.
Mapiritsi "Betacam" Masiki zviratidzo zvechirwere hypoglycemic mamiriro, akawanda acho anonzi kutyora cardiac mutinhimira. ruzivo urwu vanofanira kufunga varwere vanenge kwakakwidziridzwa ropa shuga. Ivo zvinoda kugara richiona ropa shuga yomuropa.
Kana kushandisa zvinodhaka, "Betacam" (Mahwendefa) kudzidziswa Chinyorwa anokurudzira kuteerera kudzora kwemwoyo. Kana bradycardic sinus mutinhimira zvinetso, kuti chipimo chemushonga zvakakodzera kuderedza kana kubvisa mashoko kurapwa pomutumwa.
Zvinoda nokungwarira kushandiswa kwezvinodhaka pavarwere vane dzidzo pheochromocytoma.
Tikafunga mishonga pamwe zvinoreva kuti inhalation yokutindivadza rinoitwa, chinokonzera kuora mwoyo pamusoro myocardial hunoshamisa kushanda tsandanyama uye BP. Non-depolarizing tsandanyama relaxants kuratidza munhu kwenguva refu chiito Mahwendefa apo pachena kuti "Betacam".
Kana uchida kuita munhu akaronga kuvhiya kupindira hunhu, kugadzirira kukanzura mazuva maviri asati chiitiko kuti mahwendefa havana kukanganisa zvavo yokutindivadza.
Medicament vanorega kurapwa "Betacam" mirayiridzo Chinyorwa anokurudzira kwete kamwe, asi zvishoma nezvishoma, pamwe zvinoderedza dosing 7 kana 14 days, kudzivisa maitiro muviri kuti zvinodhaka kukanzura. Ose mazuva matatu chitsama zvinodhaka ipfupi ne 0,005 d
Mahwendefa haana kubatwa zvinodhaka kuti vari retarders Monoamine oxidase enzayemu.
Hypotensive zviito zvinodhaka uye kuderedza inonzi estrogen nonsteroidal mishonga antiinflammatory izvo kutadzisa kuti yavaibvisa ions uye mvura, asi tunodzivisa kwetunhu prostaglandin yeimwe mu neitsvo.
Mawa kushandiswa diltiazem, amiodarone, uye verapamil mapiritsi "Betacam" kunotungamirira vawedzere inhibitory chiito betaxolol hydrochloride pamusoro myocardial hunoshamisa tsandanyama contractility wayo conductivity.
Tikafunga mishonga pamwe cardiac zvinodhaka glycosidic kunosimudzira atrioventricular nechigumbuso mhando.
Pamwe nemamwe antihypertensives anowedzera hypotensive basa Mahwendefa "Betacam".
Kokeini kwakaderedza kuchirapa efficacy pamusoro betaxolol zvavo mawa yaitonga.
Tikafunga "Betacam" Mahwendefa agonists kana xanthines kunokonzera yakawiriranwa kwakaderera basa ravo.
Phenothiazines uye betaxolol hydrochloride kuburikidza zvokuverengera kuwedzera kugutsikana yaro ropa.
Medicine "Betacam" kunotadzisa kubviswa kugadzirira ane lidocaine kana theophylline.
Sulfasalazine kunowedzera serum wevasungwa kuti betaxolol hydrochloride.
Hakuna mashoko kushandiswa kwezvinodhaka Varwere chiremba.
Kungwarira chinodiwa kushanda mahwendefa kuvanhu achityaira motokari, uyewo vakadzi vane pamuviri uye lactating.
Ezvemutauro izvi
By beta1-adrenoblokatornym Drug Administration classifies mushonga "Betacam" mirayiridzo Chinyorwa. Analogs uyewo nhengo kirasi iyi pharmacotherapeutic. Ane basa chirungiso mabasa sezvo betaxolol hydrochloride.
French anonzi ane analoginen zvinodhaka "Lokren", zvinoberekwa "Sanofi Winthrop Industry" muchimiro pahwendefa zvemapuranga chena firimu. Kuumba akavapotedza pamwe biconvex zviso, umo ngozi riri nokuparadzanisa Mabhuku eBraille rokuti "KE 20".
Pane imwe dose pamusoro 0.02 g betaxolol hydrochloride. Ebetsero zvinoriumba mishonga zvinosanganisira mukaka shuga, microcrystalline cellulose, yavaibvisa carboxymethyl A mhando, colloidal nesilicon dioxide, magnesium stearate.
The firimu bemhapemha sezvamunoita anogona kuonekwa hypromellose, polyethylene glycol mucherechedzo 400, titanium dioxide.
Drug kutengeswa makadhibhokisi packs it pamwe Maronda akasiyana maviri mahwendefa 14.
Ndikarangarira mushonga kubvisa BP, zviri kubatanidzwa nemamwe zvinodhaka pamusoro neBP.
The mushonga vangaita matanho kugadzirisa exacerbation kuti angina ari nerongo chimiro.
Russian nzira yakafanana iri chinodhaka "Betaxolol", iro zvinoberekwa "Moscow kwemakemikari anobudiswa chirimwa" muchimiro mahwendefa chena firimu zvemapuranga. Vane kumativi chimiro pamwe biconvex zviso. The rinoita chirungiso ichaongororwa betaxolol hydrochloride mune imwe mari 0,020 d The hwebetsero zvinoriumba zvinosanganisira mukaka shuga, yavaibvisa starch glycolate, tasara tisina mvura aerosil, magnesium stearate, microcrystalline cellulose mhando. The firimu bemhapemha chakaumbwa polyvinyl doro yakasviba-titanium, talc, Macrogol 3350 muchiso, Opadry chena-2.
chokushandisa ichi chinoshandiswa systemically pamwe cheBP.
Pane imwe mishonga "" Betaxolol "muchimiro ziso madonhwe, ayo anechekuita topically mune chirwere yakavhurika-angled yemaziso mhando dzakakwirira intraocular kumanikidzwa, kudzorera chiono pashure Laser trabekuloplasticheskogo kupindira.
pfungwa wevarwere
About rinoreva "Betacam" mirayiridzo kushandiswa varwadziwe wongororo zvinosanganisira chikamu "nenjodzi". Zviratidzo izvi vangasava kuitika kana uchishandisa mushonga.
Varwere vakawanda anogona kunzwika nyaya dzinovaka pamusoro beta1-adrenoblokatornom rinoreva "Betacam" kuti zvakakwana anobata neBP uye angina. Kumboda kutora mapiritsi pamwe chete nemamwe zvinodhaka antihypertensive mune kunzwisisa kurapa kuti mukubudirira kwavo.
Post kurapwa BP rinodzokera dzose, izvo inovandudzika zvikuru utano murwere.
Panewo wongororo zvinodhaka kuti inoratidza ineffectiveness kurapwa pamwe mumiririri uyu.
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