UtanoGadziriro

The mushonga "Spitomin": mirayiridzo kushandiswa, zviratidzo, contraindications

Nhasi isu kwamuri pamusoro zvinodhaka ichi, sezvo "Spitomin". Mirayiridzo yokushandisa, mutengo, ongororo, analogs uye mamiriro ayo - zvose nguva idzi varwere vanofarira kuti chiremba akamuraira mishonga iyi. mashoko ose anodiwa anogona kuwanikwa gare gare munyaya ino.

Description of chinodhaka, ayo chimiro, uye Zvinoumba kavha

Chii chinodhaka "Spitomin"? Mirayiridzo dzokushandisa (akatsanangura gadziriro iripo chinopiwa zvakawanda) anoti piritsi iri chena odorless, dzeraundi uye sandara chimiro, aine chamfer uye Valium uye achiita zvokutemera «E151».

The chishandiso chine buspirone hydrochloride uye ebetsero zvinoriumba zvakadai carboxymethyl starch, lactose monohydrate, magnesium stearate, yavaibvisa, microcrystalline cellulose uye colloidal anhydrous silica.

In yavakatengesa zvinodhaka paanouya mhoni packs it uye makatoni.

musimboti oparesheni

Zvii zviripo nokuda zvinodhaka "Spitomin"? Mirayiridzo dzokushandisa (Mahwendefa mutengo vakaisawo pazasi) anoti ichi anxiolytic mumiririri, iyo inesungano isiri benzodiazepine dzakatevedzana uye ane antidepressant nomugumisiro.

Kusiyana nevamwe anxiolytics, mushonga uyu haana antiepileptic, kunyaradza, hypnotic uye myorelaxant zvivako. Pfungwa dzacho kushanda inobva migumisiro buspirone ari dopaminergic uye serotonergic enyika.

Izvi zvinoreva zvokusarudza rakavhara dopamine receptors (presynaptic) uye anowedzera mwero excitation pamusoro Tutsinga tunofambisa mashoko utwu (dopamine) midbrain.

Ndezvipi zvimwe zvivako kuri muna zvinodhaka "Spitomin"? Mirayiridzo dzokushandisa inoti Buspirone ari kusarudza haasaruri agonist of 5-HT1A kweserotonin receptors. Hazvina chokuita nokusungwa benzodiazepine receptors neGhebha, uye asingadi kukanganisa psychomotor nerevane haakonzeri shiviriro. Uyezve, chokushandisa ichi hazvirevi potentiate migumisiro doro.

The kuchirapa zvinokonzerwa vaiona zvinodhaka hwapedyo zvishoma uye kunoitika pashure rimwe kana maviri pashure kurapwa.

Kinetics mari

Absorção de Água zvinodhaka "Spitomin", mirayiridzo kushandiswa riri pasi apa, rinowanikwa muna nemudumbu. Buspirone ari nezvo rinoita panguva ndima achishandisa chiropa. bioavailability wayo 4% uye kufadza yeplasma wevasungwa zvasvika pashure awa rimwe.

Buspirone ukasunungurwa pamwe mukaka. Nokuti mashoko pamusoro kupinda zvinodhaka kuburikidza placental chipingamupinyi inoshayikwa.

Kugadzirira Rinobva faeces kwemaawa mashanu.

umboo

Kubva zvaanoda "Spitomin" piritsi? Mirayiridzo kushandiswa anoratidza zvinotevera zvairatidza:

  • autonomic dysfunction chirwere;
  • kufunganya nyonganyonga iri generalized;
  • WIthdrawal chirwere doro (sezvo adjuvant kurapa);
  • tidzikame nyonganyonga ;
  • zvokuora mwoyo (sezvo adjuvant kurapa).

Contraindications

Mune zvimwe zviitiko, haisi varumbidzwa kushandisa mapiritsi "Spitomin"? Mirayiridzo yokushandisa rinoti zvinotevera pathologies uye mamiriro pasi izvo dose mishonga iri contraindicated mu:

  • yemaziso;
  • hypersensitivity kuti zvokubikisa zvinodhaka;
  • myasthenia gravis;
  • renal insufficiency, yakanyanya;
  • kuduku zera;
  • mawa negashiro Mao FIs ;
  • lactation;
  • panguva yepamuviri.

With kutarisira mumiririri chinotarisirwa mu chiropa cirrhosis uye renal kukundikana.

Medicament "Spitomin": mirayiridzo kushandiswa

Analogs zvinodhaka zvichakurukurwa pazasi.

Of mari kubatwa imwe nguva zuva, asati kana shure kudya.

The mushonga chinorambidzwa kushandisa pano neapo (ari kudiwa) kuti kurapa mwoyo, sezvo kwayo kuchirapa kushanda hwapedyo chete pashure akadzokorora kushandiswa.

The chipimo chemushonga mishonga iyi anosarudzwa nomumwe. Kazhinji, ndizvo 15 MG. Zvinofanira kukamurwa 2-3 mishonga.

Kufadza kuroorwa dose ndiyo 30 MG uye kufadza nezuva - 60 MG.

Vakwegura kugadziridzwa kuti dose runodiwa. Kana havachanyatsogoni renal kana hepatic medicament anofanira kushandiswa nokungwaririra mune mishonga diki.

nemishonga

Kazhinji mishonga "Spitomin" zvakanaka zvaitombova. Chete dzimwe nguva, chokushandisa ichi ndechechokwadi kutyorwa:

  • bhokisi marwadzo, hope, kufenda, dzungu, hypotension, nomusoro, BP;
  • huta kufunganya, chepfungwa kweropa zvirwere, dysphoric siyana, decompensation nomwoyo kukundikana, vakawedzera aikanganiswa ruzha, myocardial infarction, dysphoria, cardiomyopathy, kuzviuraya, bradycardia;
  • depersonalization, kutonhora kusashivirira, euphoria, claustrophobia, hyperkinesis, tinnitus, kufunganya, kuvaviwa mumaziso, lethargy, ziso akatsvuka, aone zvinhu zvisipo, chokundandama, kuvhiringidzika, pfungwa zvirwere;
  • madzerere, laryngitis, conjunctivitis, kuzvimba nasal mucosa, havachanyatsogoni kuravira, kunzwa Kutambudzika mubhokisi, womukati nzeve zvirwere, hyperventilation, marwadzo ziso, kushaya mhepo, photophobia, epistaxis, vakawedzera intraocular kumanikidzwa;
  • galaktoreyu, kuda kurutsa, kukuvara thyroid, flatulence, usiku enuresis, kudya kudya kuwedzera, dysuria, salivation, kumwedzi zvirwere, intestinal ropa, kunonoka ejaculation nezvimwe.

Price, analogues, wongororo

Mari mumiririri uyu 600 rubles. Kana waida, zvinonzi yakatsiva ane analoginen akadai "Buspirone Sandoz."

Consumer ongororo kukuzivisai kuti mushonga mu mubvunzo wakanaka anxiolytic mumiririri. Zvisinei, izvozvo zvinogona kutora chete nyanzvi chinangwa kwenguva refu (kwete neapo).

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