The mushonga "Buserelin Long" chinhu chakaita zvokugadzirwa analogue zvakasikwa kemikari GnRH. Kushanda ari mudziyo uri zvakananga nemakwikwi kunyorerana kuti receptors pituitary masero kwaizotevera zvinopfuura kuwedzera kwevari dzepabonde steroids mu plasma, iyo pakupedzisira kunoita zvizere blockage paiya inonzi gonadotropic pituitary chaitika. Somugumisiro mushonga "Buserelin Long" anopiwa zvakananga kudzvanyirira kemikari usage ari gonads, iyo inoratidza pacharo sezvo vasanyanye testosterone yomuropa (indices kuposita-castration) nevanhu uye kuderedza ropa estradiol kuposita-kuenda kumwedzi unhu varwere vechikadzi. Muchiitiko chokutanga tinogona kutaura pharmacological castration, yechipiri - iri postmenopausal kana ovariectomy.
The mushonga asunungurwa pakarepo somunhu lyophilizate akanyorerwa kugadzirira slurry. The Zvinoumba gadziriro ino sezvo panozogadzirika Kufananidzira zvinosanganisira anenge 4 MG buserelin acetate. Ebetsero zvinoriumba zvinosanganisira carmellose yavaibvisa, mumwe copolymer kuti glycolic uye KE-lactic acid, polysorbate-80 uye d-mannitol.
Panyaya yokushandisa zvinodhaka, yakatarwa mumiririri "Buserelin Long" nokuti mishonga kenza yemazamu uye kemikari-nemataundi kenza yeprostate. Uyezve, mushonga uyu anogona kushandiswa panguva nokurapa endometriosis. Nokuti kurapa uterine fibroids uye kushaya mbereko (kuburikidza IVF chirongwa) kunofanira kutanga kushandisa zvinodhaka "Buserelin-Long". Reviews vanachiremba apupurire migumisiro kushandiswa kwayo nokuda pakurapa endometrial hyperplastic pezvakaitwa zvakanaka.
Kana isu nezvazvo huru contraindications kushandisa, ipapo kushandisa mishonga iyi zvachose contraindicated vanhu vane nomumwe kusashivirira buserelin acetate, uyewo mamwe kwayo kutsigira zvinoriumba. Uyezve, contraindications zvinosanganisira nepamuviri uye lactation.
Oga, zvinofanira akati pamusoro zvaibvira divi migumisiro kushandisa mari "Buserelin-Long", sezvo zvinogona Somuenzaniso, mhaka urticaria, angioneurotic edema uye hyperemia. Uyezve, pangava ezvinhu akadai demineralization, hope nenyonganiso, kutemwa uye kuora mwoyo. Varwere munhukadzi kuona abdominal kurwadziwa, kuchinja libido, yakawedzera vangadikitira, menstrualnopodobnye ropa uye kuoma ari kusangana nekutsi kwemukadzi mucosa nokuda kushandisa chakaita zvokugadzirwa zvinodhaka "Buserelin-Long". Marwadzo nevanhu Anonyanyowanika chokuita exacerbation pamusoro zvinokonzera chirwere, Urinary chengetedzo, gynecomastia, uye "itsvo kuzvimba." Uyezve, unogona akacherekedza kuderera potency, yakawedzera vangadikitira, tsandanyama kusimba wamativi uye mapfupa marwadzo. A vashoma varwere tinganetseka siyana zvakadai chemanyoka zvinetso , uye pulmonary embolism.